GBR-12935 HCl - CAS# 67469-81-2 Catalog No.:M7140-2 5S)-4-((S)-N

5S)-4-((S)-N

and 30 μM

Beguinot F

12 hours) shows near complete AR degradation (>98%) in prostate cancer cells

GBR-12935 HCl - CAS# 67469-81-2 Catalog No.:M7140-2 5S)-4-((S)-NGBR 12935 HCl, CAS No. 67469 81 2, is a piperazine derivative which is a potent and selective dopamine reuptake inhibitor. It was originally developed in its 3H radiolabelled form for the purpose of mapping the distribution of dopaminergic neurons in the brain by selective labelling of dopamine transporter proteins. This has led to potential clinical uses in the diagnosis of Parkinson's disease, although selective radioligands such as Ioflupane (I)